SCHEMBL7092547

SCHEMBL7092547

CC(C)(C)OC(=O)NC1CCN(c2nc3c(cc2F)c(=O)[nH]c(=O)n3C2CC2)C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EEF2K O00418 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OGFRL1 Q5TC84 1/20 0.41
TRPV1 Q8NER1 2/20 0.41
PDE10A Q9Y233 2/20 0.41
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
SUV39H2 Q9H5I1 9/20 0.39
PARP1 P09874 1/20 0.39
BTK Q06187 1/20 0.38
CKS1B P61024 1/20 0.38
SKP1 P63208 1/20 0.38
SKP2 Q13309 1/20 0.38
AURKA O14965 1/20 0.38
PDPK1 O15530 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649040 1.00 EEF2K (0.42) EEF2KOPRM1OPRD1OPRK1OGFRL1
SCHEMBL6673219 0.86 EEF2K (0.40) EEF2KOPRM1OPRD1OPRK1OGFRL1
SCHEMBL6673221 0.86 EEF2K (0.40) EEF2KOPRM1OPRD1OPRK1OGFRL1
SCHEMBL4513304 0.85 OPRM1 (0.42) OPRM1OPRD1OPRK1OGFRL1TRPV1
SCHEMBL6674047 0.82 PIM1 (0.40) OPRM1OPRD1OPRK1OGFRL1PIM1
SCHEMBL6674052 0.82 PIM1 (0.40) OPRM1OPRD1OPRK1OGFRL1PIM1
SCHEMBL10389874 0.79 DPP4 (0.54)
SCHEMBL10389873 0.79 DPP4 (0.54)
SCHEMBL10390706 0.79 DPP4 (0.54)
SCHEMBL7093644 0.77 PIM1 (0.40) TRPV1PIM1PIM3PIM2SUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030114666-A1 Having quinazolindione core structure; non-antibiotic resistance WARNER-LAMBERT COMPANY 2003-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114666-A1 Having quinazolindione core structure; non-antibiotic resistance ABCC1, RPS6KA1, SIGMAR1 EEF2K 700/4885OPRM1 906/4885OPRD1 291/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.