SCHEMBL7092880

SCHEMBL7092880

O=C(O)C1=CC=CC=CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
THRB P10828 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
KMT2A Q03164 1/20 0.39
GABRR1 P24046 2/20 0.30
SLC6A1 P30531 1/20 0.30
SLC6A13 Q9NSD5 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL890924 0.90
SCHEMBL28256185 0.88 TSHR (0.34) TSHRMAPK1HSD17B10TDP1THRB
SCHEMBL28427720 0.88 TSHR (0.42) TSHRMAPK1HSD17B10TDP1THRB
SCHEMBL28172352 0.88
SCHEMBL28171680 0.88
Azepane SCHEMBL28329112 0.85 TSHR (0.34) TSHRMAPK1HSD17B10TDP1THRB
SCHEMBL11475296 0.81
SCHEMBL27647169 0.79 TSHR (0.35) TSHRMAPK1HSD17B10TDP1THRB
SCHEMBL11488587 0.79
Bicarbonate SCHEMBL11493509 0.77 CHRM3 (0.37) TSHRHSD17B10THRBBLMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0011670-A2 Cycloheptatriene derivatives and process for their preparation BAYER AG (DE) 1980-06-11 EP claimed
CN-106459002-B Biaryl compounds useful in the treatment of human oncological, neurological and immunological diseases 比奥根MA公司 2018-08-21 CN disclosed
CN-107699581-A 3,7 dihydroxy Zhuo phenolic ketone biological synthesis gene clusters and its application 上海交通大学 2018-02-16 CN disclosed
US-6660863-B2 Reacting an cycloheptatriene nitrile compound with nortropane compound NIHON MEDI-PHYSICS CO., LTD. (JP) 2003-12-09 US disclosed
US-6596868-B2 Reacting a cycloheptatriene derivative with a primary amine or ammonia in the presence of a base NIHON MEDI-PHYSICS CO., LTD. (JP) 2003-07-22 US disclosed
US-20030109708-A1 Process for synthesizing anhydroecgonine derivative NIHON MEDI-PHYSICS CO., LTD. 2003-06-12 US disclosed
US-20010020096-A1 Process for synthesizing anhydroecgonine derivative NIHON MEDI-PHYSICS CO., LTD. (JP) 2001-09-06 US disclosed
EP-1127887-A1 Process for synthesizing anhydroecgonine derivative NIHON MEDI-PHYSICS Co., Ltd. (JP) 2001-08-29 EP disclosed
CN-1054601-A Azabicyclo and azepine cyclic oximes and amine cholinergic agents thing and methods of treatment thereof WARNER LAMBERT CO (US) 1991-09-18 CN disclosed
EP-0011670-A3 CYCLOHEPTATRIENE DERIVATIVES AND PROCESS FOR THEIR PREPARATION BAYER AG (DE) 1980-08-20 EP disclosed
EP-0011670-A2 Cycloheptatriene derivatives and process for their preparation BAYER AG (DE) 1980-06-11 EP disclosed
EP-0011670-A2 Cycloheptatriene derivatives and process for their preparation BAYER AG (DE) 1980-06-11 EP disclosed
EP-0011669-A1 Cycloheptatriene compounds and process for the preparation of cycloheptatriene compounds BAYER AG (DE) 1980-06-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030109708-A1 Process for synthesizing anhydroecgonine derivative CES2, NPR1, OPRL1 TSHR 3513/4885MAPK1 842/4885HSD17B10 462/4885
US-20010020096-A1 Process for synthesizing anhydroecgonine derivative CES2, NPR1, OPRL1 TSHR 3513/4885MAPK1 842/4885HSD17B10 462/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.