SCHEMBL7097157

SCHEMBL7097157

CC(NC(=S)Nc1ccc(Br)cn1)n1cccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
RAB9A P51151 5/20 0.44
NPC1 O15118 4/20 0.44
POLB P06746 3/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 4/20 0.44
LTC4S Q16873 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TP53 P04637 2/20 0.41
MAPK1 P28482 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
FDPS P14324 1/20 0.40
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7579004 0.81 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL6229771 0.80 ALDH1A1 (0.48) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL8197938 0.78 TSHR (0.52) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL6805540 0.77 ALDH1A1 (0.45) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL6804222 0.76 ALDH1A1 (0.42) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL7751110 0.74 ALDH1A1 (0.54) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL6963003 0.74 ALDH1A1 (0.54) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL8197608 0.73 RAB9A (0.56) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL30557772 0.72 ALDH1A1 (0.48) ALDH1A1RAB9ANPC1POLBLMNA
SCHEMBL7749825 0.72 ALDH1A1 (0.48) ALDH1A1RAB9ANPC1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194427-B1 THIOPHENE-ETHYL THIOUREA COMPOUNDS AND USE IN THE TREATMENT OF HIV PARKER HUGHES INST (US) 2003-03-05 EP disclosed
US-6124324-A AN ENZYME INHIBITOR OF REVERSE TRANSCRIPTASE FOR THE TREATMENT OF HIV INFECTION, INCLUDING MUTANT, DRUG-SENSITIVE, DRUG-RESISTANT, AND MULTI-DRUG RESISTANT STRAINS OF HIV HUGHES INSTITUTE (US) 2000-09-26 US disclosed