SCHEMBL7097482

SCHEMBL7097482

C[C@@H](Cc1ccc(Cl)c(Cl)c1)C(=O)NC1N=C(c2ccccc2)c2ccccc2N(CC(=O)NCCN(C)C)C1=O

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OXTR P30559 13/20 0.68
PSEN1 P49768 4/20 0.53
PSEN2 P49810 4/20 0.53
APH1B Q8WW43 4/20 0.53
NCSTN Q92542 4/20 0.53
APH1A Q96BI3 4/20 0.53
PSENEN Q9NZ42 4/20 0.53
CCKBR P32239 2/20 0.52
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6005683 1.00 OXTR (0.68) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005069 0.87 OXTR (0.68) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005661 0.86 OXTR (0.70) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6003636 0.86 OXTR (0.65) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005694 0.85 OXTR (0.60) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6003771 0.82 CCKBR (0.68) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005678 0.79 OXTR (0.56) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005007 0.77 PSEN1 (0.64) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6006404 0.77 PSEN1 (0.78) OXTRPSEN1PSEN2APH1BNCSTN
SCHEMBL6005723 0.77 PSEN1 (0.65) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294702-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LTD. (GB) 2003-03-26 EP disclosed
WO-2001090084-A1 BENZODIAZEPINE DERIVATIVES AS APP MODULATORS MERCK SHARP & DOHME LIMITED (GB) 2001-11-29 WO disclosed