SCHEMBL7098503

SCHEMBL7098503

CCOc1cc([C@H]2CCN(NC)C2)cnc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.40
CHRNA4 P43681 3/20 0.40
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CHRNB4 P30926 2/20 0.32
CHRNA3 P32297 2/20 0.32
CCR5 P51681 1/20 0.31
MAPT P10636 2/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
ALK Q9UM73 1/20 0.31
TRPC6 Q9Y210 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098317 1.00 CHRNB2 (0.40) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7102514 0.93 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7103804 0.93 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7103730 0.92 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7101803 0.92 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7098388 0.88 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7103751 0.88 CHRNB2 (0.41) CHRNB2CHRNA4KDM4EALDH1A1HPGD
SCHEMBL7098864 0.80 CHRNB2 (0.35) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL7099165 0.80 PARP1 (0.31)
SCHEMBL7492241 0.80 PARP1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed