SCHEMBL7100294

SCHEMBL7100294

O=C(Nc1cccnc1)c1ccc2cccccc1-2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.68
NPC1 O15118 3/20 0.68
RAB9A P51151 3/20 0.68
LMNA P02545 2/20 0.68
GAA P10253 1/20 0.68
ALDH1A1 P00352 3/20 0.65
CHRNB2 P17787 1/20 0.65
CHRNB4 P30926 1/20 0.65
CHRNA3 P32297 1/20 0.65
CHRNA4 P43681 1/20 0.65
KMT2A Q03164 4/20 0.61
MEN1 O00255 3/20 0.61
KDM4E B2RXH2 1/20 0.61
HPGD P15428 1/20 0.61
CYP11B2 P19099 2/20 0.59
MAPT P10636 2/20 0.58
GSK3A P49840 1/20 0.58
GSK3B P49841 1/20 0.58
SORT1 Q99523 1/20 0.56
HTT P42858 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6774617 0.96 CHRNB2 (0.71) NAMPTNPC1RAB9ALMNAGAA
SCHEMBL6631304 0.85 CHRNB2 (0.89) LMNAGAAALDH1A1CHRNB2CHRNB4
SCHEMBL7020626 0.84 ALDH1A1 (0.91) GAAALDH1A1CHRNB2CHRNB4CHRNA3
SCHEMBL13948995 0.81 ALDH1A1 (0.70) NAMPTNPC1RAB9ALMNAGAA
SCHEMBL1017796 0.80 CHRNB2 (1.00) LMNAGAAALDH1A1CHRNB2CHRNB4
SCHEMBL18132518 0.79 ALDH1A1 (0.72) NAMPTNPC1RAB9ALMNAGAA
SCHEMBL6779138 0.79 ALDH1A1 (1.00) GAAALDH1A1CHRNB2CHRNB4CHRNA3
SCHEMBL7022703 0.79 CHRNB2 (0.66) NPC1RAB9ALMNAGAAALDH1A1
Hydrochloric Acid SCHEMBL29598779 0.78 CHRNB2 (0.96) LMNAGAAALDH1A1CHRNB2CHRNB4
SCHEMBL167081 0.77 NAMPT (1.00) NAMPTNPC1RAB9ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1325006-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABA A? RECEPTOR NEUROGEN CORPORATION (US) 2003-07-09 EP claimed
WO-2002012442-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABAA RECEPTOR NEUROGEN CORPORATION (US) 2002-02-14 WO claimed