SCHEMBL7100320

SCHEMBL7100320

CCC(CC(=O)NC(=O)NNC(CC(=O)O)c1ccccc1)NC(=N)N

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
ITGB3 P05106 9/20 0.42
ITGA2B P08514 8/20 0.42
ITGAV P06756 3/20 0.41
ITGB5 P18084 1/20 0.41
ITGB6 P18564 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TACR3 P29371 3/20 0.37
CTSA P10619 1/20 0.37
TACR2 P21452 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102257 0.91 KMT2A (0.42) LMNAITGB3ITGA2BITGAVCTSA
SCHEMBL7099318 0.82 ITGB3 (0.42) ITGB3ITGA2BITGAVITGB5ITGB6
SCHEMBL7100316 0.80 ITGB3 (0.39) ITGB3ITGA2BITGAVITGB5ITGB6
SCHEMBL7261894 0.77 S1PR3 (0.46) ITGB3ITGA2BITGAVITGB5ITGB6
SCHEMBL7099303 0.74 KDM4E (0.43) LMNAITGB3ITGA2BITGAVITGB5
SCHEMBL11400562 0.74 ITGB3 (0.58) ITGB3ITGA2BITGAVITGB5ITGB6
SCHEMBL7099324 0.73 ITGB3 (0.41) LMNAITGB3ITGA2BITGAVALDH1A1
SCHEMBL7099306 0.71 ITGB3 (0.51) ITGB3ITGA2BITGAVALDH1A1
SCHEMBL7102252 0.71 ITGB3 (0.39) LMNAITGB3ITGA2BITGAVCTSA
SCHEMBL17234581 0.71 ITGB3 (0.38) LMNAPOLBITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed
EP-1194401-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001005753-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2001-01-25 WO disclosed