SCHEMBL7102252

SCHEMBL7102252

CCCC(NC(=N)N)C(=O)NC(=O)NNC(CC(=O)O)c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.39
ITGAV P06756 2/20 0.39
ITGA2B P08514 2/20 0.39
CYP26A1 O43174 2/20 0.38
KMT2A Q03164 3/20 0.37
CTSA P10619 3/20 0.37
GABBR2 O75899 3/20 0.35
GABBR1 Q9UBS5 3/20 0.35
CYP2C9 P11712 3/20 0.35
LMNA P02545 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 2/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
NFKB1 P19838 1/20 0.35
DRD3 P35462 1/20 0.35
BLM P54132 1/20 0.35
CYP1A2 P05177 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7100316 0.91 ITGB3 (0.39) ITGB3ITGAVITGA2BCYP2C9CYP2D6
SCHEMBL7261894 0.82 S1PR3 (0.46) ITGB3ITGAVITGA2BKMT2ACTSA
SCHEMBL7102257 0.81 KMT2A (0.42) ITGB3ITGAVITGA2BCYP26A1KMT2A
SCHEMBL7099318 0.74 ITGB3 (0.42) ITGB3ITGAVITGA2BCTSA
SCHEMBL7104747 0.73 CTSA (0.42) ITGB3ITGAVITGA2BCYP26A1KMT2A
SCHEMBL7103319 0.73 ITGB3 (0.46) ITGB3ITGAVITGA2BKMT2ACTSA
SCHEMBL7104753 0.71 ITGB3 (0.51) ITGB3ITGAVITGA2BKMT2ACTSA
SCHEMBL7100320 0.71 LMNA (0.42) ITGB3ITGAVITGA2BCTSALMNA
SCHEMBL7261904 0.69 KMT2A (0.41) ITGB3ITGAVITGA2BKMT2ACTSA
SCHEMBL7099303 0.65 KDM4E (0.43) ITGB3ITGAVITGA2BKMT2ACTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed