SCHEMBL7100343

SCHEMBL7100343

CCOC(=O)C(C)c1ccc(-n2c(CC)nc3cc(C#N)c(Cl)cc32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP11B2 P19099 1/20 0.35
MAT2A P31153 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
PGK1 P00558 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HPGD P15428 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099008 0.89 SMN1; SMN2 (0.40) HTTSMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL7098251 0.85 SMN1; SMN2 (0.39) SMN1; SMN2PSEN1PSEN2APH1BNCSTN
SCHEMBL7102170 0.83 SMN1; SMN2 (0.36) SMN1; SMN2PSEN1PSEN2APH1BNCSTN
SCHEMBL7097040 0.82 ESR1 (0.40) HTTSMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL7100074 0.82 NPC1 (0.42) SMN1; SMN2PGK1ALDH1A1MAPTPOLB
SCHEMBL6426223 0.82 PSEN1 (0.45) SMN1; SMN2PSEN1PSEN2APH1BNCSTN
SCHEMBL27600113 0.82 PSEN1 (0.47) SMN1; SMN2PSEN1PSEN2APH1BNCSTN
SCHEMBL27599858 0.81 CYP1A2 (0.40) MAT2APGK1ALDH1A1MAPTHPGD
SCHEMBL7105813 0.80 ALDH1A1 (0.43) HTTSMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL1625820 0.79 AR (0.37) HTTHSD17B10CYP11B2MAT2APGK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326606-A2 EP4 RECEPTOR INHIBITORS TO TREAT RHEUMATOID ARTHRITIS PFIZER PHARMACEUTICALS INC. (JP) 2003-07-16 EP disclosed
WO-2002032422-A2 EP4 RECEPTOR INHIBITORS TO TREAT RHEUMATOID ARTHRITIS PFIZER PHARMACEUTICALS INC. (JP) 2002-04-25 WO disclosed