SCHEMBL7101243

SCHEMBL7101243

CNN1CC[C@@H](c2cnc(Cl)c(F)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 8/20 0.32
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
PARP1 P09874 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
PIK3C3 Q8NEB9 1/20 0.31
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7102509 1.00 EGLN1 (0.32) EGLN1S1PR1S1PR3PARP1CHRM2
SCHEMBL7097819 0.92 PROKR1 (0.35) HRH4HRH3
SCHEMBL7101894 0.92 PROKR1 (0.35) HRH4HRH3
SCHEMBL7105294 0.91 PROKR1 (0.36) HRH4HRH3
SCHEMBL7101818 0.91 PROKR1 (0.36) HRH4HRH3
SCHEMBL7102628 0.87 EGLN1 (0.33) EGLN1S1PR1S1PR3PARP1HRH4
SCHEMBL7098888 0.87 EGLN1 (0.33) EGLN1S1PR1S1PR3PARP1HRH4
SCHEMBL7105235 0.86 CHRNB2 (0.36) EGLN1
SCHEMBL7098850 0.86 CHRNB2 (0.36) EGLN1
SCHEMBL7097540 0.85 CHRNB2 (0.39) EGLN1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed