SCHEMBL7101818

SCHEMBL7101818

CNN1CCCC[C@@H](c2cnc(Cl)c(F)c2)C1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 8/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105294 1.00 PROKR1 (0.36) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7101894 0.96 PROKR1 (0.35) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7097819 0.96 PROKR1 (0.35) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7101243 0.91 EGLN1 (0.32) HRH4HRH3
SCHEMBL7102509 0.91 EGLN1 (0.32) HRH4HRH3
SCHEMBL7492251 0.87 SLC6A2 (0.43) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7097808 0.87 SLC6A2 (0.43) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7098418 0.86 ALDH1A1 (0.44) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7098872 0.86 SLC6A2 (0.39) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7103653 0.86 SLC6A2 (0.39) PROKR1SLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed