SCHEMBL7101379

SCHEMBL7101379

COc1cccc(OC)c1C=CC(=O)c1ccc(N)cc1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.85
CA1 P00915 2/20 0.62
CA2 P00918 2/20 0.62
KRAS P01116 1/20 0.62
CTSL P07711 1/20 0.59
CTSB P07858 1/20 0.59
MAOA P21397 2/20 0.58
CYP1A2 P05177 3/20 0.56
CYP2D6 P10635 2/20 0.56
CYP1A1 P04798 1/20 0.56
PTPN1 P18031 1/20 0.55
CYP1B1 Q16678 1/20 0.54
NPC1 O15118 2/20 0.54
LMNA P02545 2/20 0.54
MAPT P10636 2/20 0.54
BCHE P06276 1/20 0.54
RAB9A P51151 1/20 0.54
MAOB P27338 3/20 0.54
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7192430 1.00 ABCG2 (0.85) ABCG2CA1CA2KRASCTSL
SCHEMBL7185747 0.86 ABCG2 (0.88) ABCG2CTSLCTSBMAOACYP1A2
SCHEMBL7185751 0.86 ABCG2 (0.88) ABCG2CTSLCTSBMAOACYP1A2
SCHEMBL979720 0.86 ABCG2 (0.87) ABCG2MAOACYP1A2CYP2D6CYP1A1
SCHEMBL979719 0.86 ABCG2 (0.87) ABCG2MAOACYP1A2CYP2D6CYP1A1
SCHEMBL7803092 0.85 ABCG2 (0.61) ABCG2CA1CA2KRASCTSL
SCHEMBL7803088 0.85 ABCG2 (0.61) ABCG2CA1CA2KRASCTSL
SCHEMBL7096493 0.85 ABCG2 (0.70) ABCG2CA1CA2KRASMAOA
SCHEMBL7102265 0.85 ABCG2 (0.86) ABCG2CA1CA2KRASCTSL
SCHEMBL7187466 0.84 ABCG2 (0.60) ABCG2CA1CA2KRASCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003097577-A1 CHEMICAL COMPOUND CONSISTING OF A NITROGENOUS CHALCONE DERIVATIVE, METHOD OF PRODUCING ONE SUCH CHEMICAL COMPOUND AND FILTERING AND/OR COSMETIC COMPOSITION CONTAINING SAME SYNTH'E163 (SOCIETE ANONYME) (FR) 2003-11-27 WO claimed
WO-2003097577-A1 CHEMICAL COMPOUND CONSISTING OF A NITROGENOUS CHALCONE DERIVATIVE, METHOD OF PRODUCING ONE SUCH CHEMICAL COMPOUND AND FILTERING AND/OR COSMETIC COMPOSITION CONTAINING SAME SYNTH'E163 (SOCIETE ANONYME) (FR) 2003-11-27 WO disclosed
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed