SCHEMBL7101580

SCHEMBL7101580

NCCc1nc(N)nc(-c2ccc(Cl)cc2Cl)c1CN1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 3/20 0.45
SLC2A2 P11168 1/20 0.44
DPP4 P27487 9/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
AR P10275 1/20 0.39
SLC2A1 P11166 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846684 0.78 GSK3B (0.52) CYP2A13SLC2A2KDM4EALDH1A1MAPT
SCHEMBL27538115 0.76 CYP2A13 (0.55) CYP2A13SLC2A2KDM4EALDH1A1MAPT
SCHEMBL3370971 0.70 DPP4 (0.56) DPP4NPC1RAB9ACYP3A4
SCHEMBL5099299 0.69 CYP2A13 (0.48) CYP2A13SLC2A2KDM4EALDH1A1MAPT
SCHEMBL7857358 0.68 DHFR (0.49) DPP4MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL5082578 0.67 DPP4 (0.48) DPP4CYP3A4
SCHEMBL4972403 0.66 CYP2A13 (0.56) CYP2A13SLC2A2KDM4EALDH1A1MAPT
SCHEMBL3601192 0.65 TSHR (0.44) CYP2A13SLC2A2DPP4HTTSMN1; SMN2
SCHEMBL4109682 0.64 CYP2A13 (1.00) CYP2A13KDM4EALDH1A1MAPTMAPK1
SCHEMBL6068869 0.64 CYP2A13 (0.56) CYP2A13SLC2A2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed