SCHEMBL7101866

SCHEMBL7101866

CC(C)NCCCNS(=O)(=O)Nc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.42
CA12 O43570 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
POLB P06746 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
LMNA P02545 3/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
IL1RN P18510 1/20 0.37
ERAP1 Q9NZ08 1/20 0.37
CACNA2D1 P54289 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19798391 0.80 CA1 (0.55) KEAP1CA12CA7CA9CA14
SCHEMBL20724723 0.79 AR (0.45) KEAP1CA12CA7CA9CA1
SCHEMBL19798396 0.78 KEAP1 (0.42) KEAP1CA12CA9POLBCA1
SCHEMBL29124111 0.78 PPARA (0.55) CA12CA7CA9CA14CA1
SCHEMBL15444483 0.77 KEAP1 (0.42) KEAP1CA12CA7CA14POLB
SCHEMBL15592740 0.76 KEAP1 (0.46) KEAP1CA12CA7CA9CA1
SCHEMBL28044679 0.75 KEAP1 (0.48) KEAP1CA12CA7CA9CA14
SCHEMBL17199172 0.73 KEAP1 (0.47) KEAP1CA12CA7CA9CA14
SCHEMBL7835580 0.73 CA2 (0.45) KEAP1CA12CA7CA9CA14
SCHEMBL19798740 0.73 MAPK1 (0.43) KEAP1CA12CA7CA14POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303496-A1 PYRIMIDINE DERIVATIVES AstraZeneca AB (SE) 2003-04-23 EP disclosed
WO-2002004429-A1 PYRIMIDINE DERIVATIVES ASTRAZENECA AB (SE) 2002-01-17 WO disclosed