SCHEMBL7101962

SCHEMBL7101962

COc1cccc(-c2sc3ccccc3c2Oc2ccc(OCCBr)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.58
NAPEPLD Q6IQ20 1/20 0.58
HCRTR1 O43613 1/20 0.51
L3MBTL1 Q9Y468 3/20 0.44
PAX8 Q06710 1/20 0.44
ESR1 P03372 4/20 0.43
ESR2 Q92731 3/20 0.43
ATM Q13315 2/20 0.43
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42
TUBA4A P68366 1/20 0.42
TUBB4B P68371 1/20 0.42
TUBB3 Q13509 1/20 0.42
TUBB2A Q13885 1/20 0.42
TUBB8 Q3ZCM7 1/20 0.42
TUBA3E Q6PEY2 1/20 0.42
TUBA1A Q71U36 1/20 0.42
TUBA1C Q9BQE3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7106095 0.92 TUBB4A (0.51) ITGA4NAPEPLDHCRTR1L3MBTL1ESR1
SCHEMBL7106562 0.89 ITGA4 (0.58) ITGA4NAPEPLDHCRTR1L3MBTL1PAX8
SCHEMBL7108616 0.85 ITGA4 (0.51) ITGA4NAPEPLDHCRTR1L3MBTL1PAX8
SCHEMBL7106045 0.85 ITGA4 (0.53) ITGA4NAPEPLDHCRTR1L3MBTL1ESR1
SCHEMBL7101221 0.83 ESR1 (0.66) ITGA4ESR1ESR2UBE2N
SCHEMBL7108339 0.83 ESR1 (0.61) ITGA4NAPEPLDESR1ESR2ALDH1A1
SCHEMBL7101025 0.83 ITGA4 (0.51) ITGA4NAPEPLDHCRTR1L3MBTL1PAX8
SCHEMBL7101796 0.83 ESR1 (0.50) ITGA4NAPEPLDL3MBTL1ESR1ESR2
Hydrochloric Acid SCHEMBL7103199 0.82 ESR1 (0.65) ITGA4ESR1ESR2UBE2N
SCHEMBL17155697 0.82 TUBB4A (0.63) ESR1ESR2TUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827959-B1 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5977382-A Benzo[b]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
US-5977098-A Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
EP-0827959-A2 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-03-11 EP disclosed