SCHEMBL7103044

SCHEMBL7103044

N#CN=C(NCCCCCCOC(=O)c1ccc(Cl)cc1)Nc1ccncc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.59
NAMPT P43490 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 7/20 0.42
ALDH1A1 P00352 2/20 0.42
NT5E P21589 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 6/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ROCK2 O75116 2/20 0.39
RAB9A P51151 2/20 0.38
HPGD P15428 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL810378 0.87 IKBKB (0.56) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL810238 0.85 IKBKB (0.54) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL810930 0.85 IKBKB (0.54) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL811142 0.85 IKBKB (0.54) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL12083293 0.85 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8917545 0.85 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL810990 0.85 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8918236 0.85 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL16312347 0.85 IKBKB (0.80) IKBKBNAMPTCYP3A4CYP2D6CYP2C9
Chs-828 SCHEMBL7148798 0.84 IKBKB (0.79) IKBKBNAMPTCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984938-B1 CYANOGUANIDINES AS CELL PROLIFERATION INHIBITORS LEO PHARMA AS WITH SECONDARY N (DK) 2003-09-10 EP claimed
EP-0984938-B1 CYANOGUANIDINES AS CELL PROLIFERATION INHIBITORS LEO PHARMA AS WITH SECONDARY N (DK) 2003-09-10 EP disclosed