SCHEMBL810238

SCHEMBL810238

N#CN=C(NCCCCCCC(=O)c1ccc(Cl)cc1)Nc1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.54
KMT2A Q03164 3/20 0.44
NT5E P21589 1/20 0.44
NAMPT P43490 4/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MEN1 O00255 2/20 0.40
HDAC3 O15379 3/20 0.40
HDAC4 P56524 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC7 Q8WUI4 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC10 Q969S8 3/20 0.40
HDAC11 Q96DB2 3/20 0.40
HDAC8 Q9BY41 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC9 Q9UKV0 3/20 0.40
HDAC5 Q9UQL6 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL811142 1.00 IKBKB (0.54) IKBKBKMT2ANT5ENAMPTCYP2C9
SCHEMBL810930 1.00 IKBKB (0.54) IKBKBKMT2ANT5ENAMPTCYP2C9
SCHEMBL810378 0.89 IKBKB (0.56) IKBKBKMT2ANT5ENAMPTCYP2C9
SCHEMBL7103044 0.85 IKBKB (0.59) IKBKBKMT2ANT5ENAMPTCYP2C9
SCHEMBL7098728 0.83 CYP1A2 (0.53) IKBKBNAMPTCYP2C9CYP2C19HDAC3
SCHEMBL20095475 0.83 CYP1A2 (0.53) IKBKBNAMPTCYP2C9CYP2C19HDAC3
SCHEMBL8918236 0.81 IKBKB (0.80) IKBKBKMT2ANAMPTCYP2C9CYP2C19
Chs-828 SCHEMBL16312347 0.81 IKBKB (0.80) IKBKBKMT2ANAMPTCYP2C9CYP2C19
Chs-828 SCHEMBL12083293 0.81 IKBKB (0.80) IKBKBKMT2ANAMPTCYP2C9CYP2C19
SCHEMBL8917545 0.81 IKBKB (0.80) IKBKBKMT2ANAMPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394649-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDYL CYANOGUANIDINES, PREPARATION METHODS AND USES THEREOF Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2011-12-14 EP disclosed