SCHEMBL810378

SCHEMBL810378

N#CN=C(NCCCCCCNC(=O)c1ccc(Cl)cc1)Nc1ccncc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.56
NT5E P21589 1/20 0.52
KMT2A Q03164 1/20 0.52
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
NAAA Q02083 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP1A2 P05177 1/20 0.45
NAMPT P43490 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL810238 0.89 IKBKB (0.54) IKBKBNT5EKMT2AHDAC3HDAC4
SCHEMBL811142 0.89 IKBKB (0.54) IKBKBNT5EKMT2AHDAC3HDAC4
SCHEMBL810930 0.89 IKBKB (0.54) IKBKBNT5EKMT2AHDAC3HDAC4
SCHEMBL810405 0.89 CYP1A2 (0.50) IKBKBHDAC3HDAC4HDAC1HDAC7
SCHEMBL7103044 0.87 IKBKB (0.59) IKBKBNT5EKMT2ACYP2C9CYP2C19
SCHEMBL810996 0.86 PSEN1 (0.53) IKBKBKMT2AHDAC3HDAC4HDAC1
SCHEMBL6615293 0.84 CYP11B1 (0.57) KMT2AMAPK1NAMPT
Chs-828 SCHEMBL16312347 0.83 IKBKB (0.80) IKBKBKMT2AMAPK1CYP2C9CYP2C19
Chs-828 SCHEMBL12083293 0.83 IKBKB (0.80) IKBKBKMT2AMAPK1CYP2C9CYP2C19
SCHEMBL8918236 0.83 IKBKB (0.80) IKBKBKMT2AMAPK1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394649-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDYL CYANOGUANIDINES, PREPARATION METHODS AND USES THEREOF Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2011-12-14 EP disclosed