SCHEMBL7103451

SCHEMBL7103451

CNN1CCC[C@H](c2cnc(Cl)c(Cl)c2)C1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 14/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
CHRNB2 P17787 2/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
CHRNA4 P43681 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7492594 1.00 PROKR1 (0.38) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7492251 0.96 SLC6A2 (0.43) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7097808 0.96 SLC6A2 (0.43) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7105235 0.92 CHRNB2 (0.36) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7098850 0.92 CHRNB2 (0.36) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7487049 0.89 EGLN1 (0.35) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7098866 0.89 EGLN1 (0.35) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7104089 0.88 CHRNB2 (0.38) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7099348 0.88 CHRNB2 (0.38) PROKR1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7105555 0.88 ALDH1A1 (0.39) PROKR1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed