SCHEMBL7103520

SCHEMBL7103520

CC(=O)NC[C@H]1CN(c2cc(F)c(C3=CCNCC3)c(F)c2)C(=O)O1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.55
MAOB P27338 3/20 0.54
PTGS1 P23219 2/20 0.54
SDHA P31040 2/20 0.54
LMNA P02545 1/20 0.54
CALML3 P27482 1/20 0.54
F10 P00742 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103523 1.00 MAOA (0.55) MAOAMAOBPTGS1SDHALMNA
Hydrochloric Acid SCHEMBL5678891 0.88 MAOA (0.71) MAOAMAOBPTGS1SDHALMNA
Hydrochloric Acid SCHEMBL5678897 0.88 MAOA (0.71) MAOAMAOBPTGS1SDHALMNA
SCHEMBL5678811 0.88 MAOA (0.71) MAOAMAOBPTGS1SDHALMNA
SCHEMBL5678812 0.88 MAOA (0.71) MAOAMAOBPTGS1SDHALMNA
Hydrochloric Acid SCHEMBL5833975 0.85 MAOA (0.41) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6398607 0.84 MAOA (0.51) MAOAMAOBPTGS1SDHALMNA
SCHEMBL6399424 0.84 MAOA (0.51) MAOAMAOBPTGS1SDHALMNA
SCHEMBL7025191 0.84 MAOA (0.59) MAOAMAOBPTGS1SDHALMNA
SCHEMBL7691880 0.83 MAOA (0.60) MAOAMAOBPTGS1SDHALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6638955-B2 Antibiotic oxazolidinone derivatives SYNGENTA LIMITED (GB) 2003-10-28 US disclosed
US-20020133022-A1 Antibiotic oxazolidinone derivatives SYNGENTA LIMITED (GB) 2002-09-19 US disclosed
US-6365751-B1 ACTIVE AGAINST GRAM-POSITIVE BACTERIA, IN PARTICULAR, AGAINST STRAINS RESISTANT TO VANCOMYCIN, AMINOGLYCOSIDES AND PENCILLINS AND DERIVATIVES; NONTOXIC ZENECA LTD. (GB) 2002-04-02 US disclosed
US-6271383-B1 USEFUL ACTIVITY AGAINST GRAM-POSITIVE PATHOGENS; IN PARTICULAR, AGAINST VARIOUS STRAINS EXHIBITING RESISTANCE TO VANCOMYCIN AND AGAINST E. FAECIUM STRAINS RESISTANT TO BOTH AMINOGLYCOSIDES AND CLINICALLY USED BETA-LACTAMS. ZENECA LIMITED (GB) 2001-08-07 US disclosed
US-5981528-A Antibiotic oxazolidinone derivatives ZENECA LIMITED 1999-11-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020133022-A1 Antibiotic oxazolidinone derivatives OXA1L, POLN, MRPL21 MAOA 2791/4885MAOB 2698/4885PTGS1 4069/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.