SCHEMBL7103801

SCHEMBL7103801

COc1ccc(Cc2nc(-c3ccsc3)c[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
PDGFRB P09619 3/20 0.46
LTA4H P09960 1/20 0.44
RET P07949 1/20 0.43
GPBAR1 Q8TDU6 2/20 0.42
PDGFRA P16234 2/20 0.40
COMT P21964 1/20 0.39
ALOX5 P09917 1/20 0.38
CYP17A1 P05093 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14334208 0.83 RET (0.40) PDGFRBRETGPBAR1CYP17A1CYP11B1
SCHEMBL7100910 0.82 GSK3B (0.41) PDGFRBLTA4HRETCYP17A1CYP11B1
SCHEMBL6210283 0.81 LTA4H (0.51) NPC1LTA4HCYP11B1CYP11B2
SCHEMBL14334743 0.77 RET (0.43) PDGFRBRETPDGFRA
SCHEMBL14334462 0.76 PDGFRB (0.39) NPC1PDGFRBRETPDGFRACYP17A1
SCHEMBL4317092 0.74 CYP17A1 (0.60) NPC1PDGFRBLTA4HRETGPBAR1
SCHEMBL10905429 0.74 LTA4H (0.47) LTA4H
SCHEMBL14334131 0.73 MAPK1 (0.40) PDGFRBRET
SCHEMBL5758497 0.73 CASP3 (0.49) NPC1PDGFRBPDGFRA
SCHEMBL11771733 0.73 LTA4H (0.46) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500357-A 2003-01-07 JP claimed
EP-1194144-A4 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-08-07 EP claimed
EP-1194144-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-10 EP claimed
WO-2000071120-A1 ANTIBACTERIAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-11-30 WO claimed