SCHEMBL7104020

SCHEMBL7104020

COc1ccc(CNC(=O)c2cc3c(=O)n(Cc4cccc(C(=O)O)c4C(C)(C)C)c(=O)n(C)c3cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 5/20 0.48
SLC22A8 Q8TCC7 1/20 0.48
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXFP1 Q9HBX9 2/20 0.40
TP53 P04637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PPARG P37231 1/20 0.39
TSHR P16473 1/20 0.39
ASPH Q12797 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104026 0.88 MMP13 (0.48) MMP13SLC22A8KDM4EMAPK1HTT
SCHEMBL6428872 0.83 MMP13 (0.53) MMP13SLC22A8KDM4ERXFP1ALDH1A1
SCHEMBL6364247 0.83 MMP13 (0.65) MMP13SLC22A8ALDH1A1HPGDCYP1A2
SCHEMBL6295571 0.80 MMP13 (0.56) MMP13SLC22A8SMN1; SMN2RXFP1TP53
SCHEMBL6468114 0.79 MMP13 (0.67) MMP13SLC22A8TP53MAPT
SCHEMBL6256740 0.78 MMP13 (0.51) MMP13SLC22A8KDM4EMAPK1HTT
SCHEMBL7100732 0.76 PIK3CD (0.51) MMP13SLC22A8KDM4EMAPK1ALDH1A1
SCHEMBL7017009 0.72 MAPT (0.51) KDM4EMAPK1HTTSMN1; SMN2RXFP1
SCHEMBL8311521 0.72 L3MBTL1 (0.46) MMP13SLC22A8MAPK1SMN1; SMN2TP53
SCHEMBL6724659 0.71 PPARG (0.53) MMP13KDM4ERXFP1ALDH1A1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368324-A1 QUINAZOLINES AS MMP-13 INHIBITORS Warner-Lambert Company LLC (US) 2003-12-10 EP disclosed
WO-2002064572-A1 QUINAZOLINES AS MMP-13 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed