SCHEMBL7104731

SCHEMBL7104731

OC1(c2ccc(F)cc2)CCC(N2CCC(Cc3cc(F)ccc3F)CC2)CC1

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.52
CCR1 P32246 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7041180 0.88 SLC6A4 (0.59) SLC6A4
SCHEMBL7038210 0.84
SCHEMBL7040750 0.81 GRIN2B (0.53) CCR1
SCHEMBL8829509 0.78 DPP4 (0.49) SLC6A4
SCHEMBL7107899 0.76 HTR1D (0.54) SLC6A4
SCHEMBL7110814 0.75 SLC6A4 (0.57) SLC6A4
SCHEMBL7307698 0.74 HTR1D (0.53)
SCHEMBL7038215 0.73 HTR1D (0.54)
SCHEMBL7304581 0.73 CCR1 (0.48) CCR1
SCHEMBL9036819 0.73 HTR1D (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387593-A Anxiolytic agents BRISTON-MYERS SQUIBB (US) 1995-02-07 US claimed
EP-1037637-B1 USE OF 5HT1A RECEPTOR ANTAGONISTS FOR PREVENTING AND/OR TREATING TEMPORAL LOBE EPILEPSY UNIV PRINCETON (US) 2003-03-19 EP disclosed
EP-1037637-A1 USE OF 5HT1A RECEPTOR ANTAGONISTS FOR PREVENTING AND/OR TREATING TEMPORAL LOBE EPILEPSY PRINCETON UNIVERSITY (US) 2000-09-27 EP disclosed
WO-1999029323-A1 USE OF 5HT1A RECEPTOR ANTAGONISTS FOR PREVENTING AND/OR TREATING TEMPORAL LOBE EPILEPSY PRINCETON UNIVERSITY (US) 1999-06-17 WO disclosed
EP-0546583-B1 Piperazinyl-and piperidinyl-cyclohexanols BRISTOL MYERS SQUIBB CO (US) 1996-05-22 EP disclosed
US-5478828-A Anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-12-26 US disclosed
US-5387593-A Anxiolytic agents BRISTON-MYERS SQUIBB (US) 1995-02-07 US disclosed
EP-0546583-A1 Piperazinyl-and piperidinyl-cyclohexanols Bristol-Myers Squibb Company (US) 1993-06-16 EP disclosed