SCHEMBL7304581

SCHEMBL7304581

OC1(c2ccc(F)cc2)CCC(N2CCNCC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.48
OPRM1 P35372 2/20 0.43
OPRD1 P41143 2/20 0.43
OPRK1 P41145 2/20 0.43
OPRL1 P41146 2/20 0.43
POLB P06746 1/20 0.42
DRD2 P14416 1/20 0.41
RORC P51449 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036683 0.85 OPRL1 (0.45) CCR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL9036194 0.79 LIPG (0.40) CCR1OPRL1DRD2RORCHPGD
SCHEMBL7305248 0.78 HTR1D (0.57) OPRL1
SCHEMBL615480 0.77 DRD2 (0.66) OPRM1OPRD1OPRK1OPRL1DRD2
Hydrochloric Acid SCHEMBL7079664 0.76 CCR1 (0.43) CCR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL8192038 0.76 HTR1D (0.64)
Hydrochloric Acid SCHEMBL1765160 0.76 DRD2 (0.63) OPRM1OPRD1OPRK1OPRL1DRD2
SCHEMBL11594980 0.75 CCR1 (0.56) CCR1DRD2
SCHEMBL11593464 0.75 CCR1 (0.50) CCR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL7299616 0.75 HTR1D (0.66) OPRL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153611-A AS NON-DOPAMINERGIC ANTIISCHEMIC COMPOUNDS FOR TREATING BRAIN DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-11-28 US disclosed
EP-0546583-B1 Piperazinyl-and piperidinyl-cyclohexanols BRISTOL MYERS SQUIBB CO (US) 1996-05-22 EP disclosed
US-5478828-A Anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-12-26 US disclosed
EP-0560669-B1 Piperazinyl-and piperidinyl-cyclohexenes and cyclohexanes BRISTOL MYERS SQUIBB CO (US) 1995-06-14 EP disclosed
US-5387593-A Anxiolytic agents BRISTON-MYERS SQUIBB (US) 1995-02-07 US disclosed
EP-0560669-A1 Piperazinyl-and piperidinyl-cyclohexenes and cyclohexanes Bristol-Myers Squibb Company (US) 1993-09-15 EP disclosed
EP-0546583-A1 Piperazinyl-and piperidinyl-cyclohexanols Bristol-Myers Squibb Company (US) 1993-06-16 EP disclosed