SCHEMBL7104864

SCHEMBL7104864

Cc1ccc(C(=O)c2c(-c3ccc(O)cc3)sc3cc(O)ccc23)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 1.00
ESR2 Q92731 15/20 0.71
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
TDP1 Q9NUW8 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1665657 0.93 ESR1 (0.86) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL15660902 0.92 ESR1 (0.85) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL25079639 0.89 ESR1 (0.81) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8630381 0.89 ESR1 (0.80) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL26158897 0.88 ESR1 (0.79) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8628025 0.86 ESR1 (0.76) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8562371 0.86 ESR1 (0.76) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8626952 0.86 ESR1 (0.80) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL31683627 0.86 ESR1 (0.81) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8631942 0.86 ESR1 (0.81) ESR1ESR2MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819686-B1 Benzothiophene compounds, and uses and formulations thereof LILLY CO ELI (US) 2003-10-01 EP disclosed
US-5780648-A Benzothiophene compounds, and uses formulations thereof ELI LILLY AND COMPANY (US) 1998-07-14 US disclosed
EP-0819686-A1 Benzothiophene compounds, and uses and formulations thereof ELI LILLY AND COMPANY (US) 1998-01-21 EP disclosed