SCHEMBL8630381

SCHEMBL8630381

CC(=O)Oc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.80
ESR2 Q92731 10/20 0.63
MEN1 O00255 1/20 0.54
PLD2 O14939 1/20 0.54
KDM1A O60341 1/20 0.54
NR1I2 O75469 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
C5 P01031 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
FYN P06241 1/20 0.54
PGR P06401 1/20 0.54
CYP3A4 P08684 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54
ADRB3 P13945 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628025 0.93 ESR1 (0.76) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL8625838 0.92 ESR1 (0.65) ESR1ESR2LMNACNR1
SCHEMBL7104864 0.89 ESR1 (1.00) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL7075690 0.86 TUBB4A (0.60) ESR1ESR2CNR1HSD17B10
SCHEMBL11547223 0.86 ESR1 (0.63) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL15660902 0.84 ESR1 (0.85) ESR1ESR2MEN1KMT2ATDP1
SCHEMBL8340581 0.84 ESR1 (0.74) ESR1ESR2LMNA
SCHEMBL7075381 0.84 ESR1 (0.72) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11548512 0.83 CNR1 (0.71) ESR1ESR2CNR1TDP1
SCHEMBL7075664 0.83 ESR1 (0.74) ESR1ESR2MEN1PLD2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780648-A Benzothiophene compounds, and uses formulations thereof ELI LILLY AND COMPANY (US) 1998-07-14 US disclosed