SCHEMBL7105191

SCHEMBL7105191

COc1ccc(C(CC(=O)O)CC(=O)NNC(=O)c2cccc(NC(=N)N)c2)cc1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.69
ITGAV P06756 17/20 0.69
ITGA2B P08514 3/20 0.54
FNTA P49354 2/20 0.50
FNTB P49356 2/20 0.50
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104776 0.91 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL13703191 0.89 ITGB3 (0.57) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7099298 0.89 ITGB3 (0.66) ITGB3ITGAVITGA2B
SCHEMBL7104742 0.87 ITGB3 (0.68) ITGB3ITGAVITGA2B
SCHEMBL7105309 0.87 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7102231 0.87 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7099697 0.87 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7103664 0.83 ITGB3 (0.68) ITGB3ITGAVITGA2B
SCHEMBL7105186 0.82 ITGB3 (0.57) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7106602 0.80 ITGB3 (0.67) ITGB3ITGAVITGA2BFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed
EP-1194401-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001005753-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2001-01-25 WO disclosed