SCHEMBL7099697

SCHEMBL7099697

N=C(N)Nc1cccc(C(=O)NNC(=O)CC(CC(=O)O)c2ccc(Br)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 18/20 0.68
ITGAV P06756 17/20 0.68
ITGA2B P08514 5/20 0.55
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099298 0.92 ITGB3 (0.66) ITGB3ITGAVITGA2BHTTSMN1; SMN2
SCHEMBL7106602 0.90 ITGB3 (0.67) ITGB3ITGAVITGA2BHTTSMN1; SMN2
SCHEMBL7102231 0.90 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7105309 0.90 ITGB3 (0.68) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7104742 0.90 ITGB3 (0.68) ITGB3ITGAVITGA2B
SCHEMBL13703191 0.90 ITGB3 (0.57) ITGB3ITGAVITGA2BHTTSMN1; SMN2
SCHEMBL7105191 0.87 ITGB3 (0.69) ITGB3ITGAVITGA2BFNTAFNTB
SCHEMBL7103664 0.86 ITGB3 (0.68) ITGB3ITGAVITGA2B
SCHEMBL7099030 0.82 ITGB3 (0.52) ITGB3ITGAVITGA2B
SCHEMBL7098907 0.80 ITGB3 (0.67) ITGB3ITGAVITGA2BHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed
EP-1194401-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001005753-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2001-01-25 WO disclosed