SCHEMBL7105344

SCHEMBL7105344

CC1(C)[C@@H](C(=O)N[C@@H](Cc2ccc(OCc3c(Cl)cccc3Cl)cn2)C(=O)O)CC[C@]1(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 19/20 0.47
ITGB1 P05556 2/20 0.46
ITGB3 P05106 1/20 0.46
ITGAV P06756 1/20 0.46
ITGA5 P08648 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098651 0.94 MEN1 (0.42) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL7102227 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7102228 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7098304 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7098069 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7098305 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7242947 0.88 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7228642 0.87 ITGA4 (0.42) ITGA4ITGB1
SCHEMBL7103946 0.84 ITGA4 (0.39) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL6561139 0.84 ITGA4 (0.49) ITGA4ITGB1ITGB3ITGAVITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991619-B1 INHIBITORS OF ALPHA 4-BETA 1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2003-09-10 EP disclosed
US-6596752-B1 Small molecules that are potent inhibitors of alpha 4 beta 1 mediated adhesion to either VCAM or CS-1 and which could be useful for the treatment of inflammatory diseases. TANABE SEIYAKU CO., LTD. (JP) 2003-07-22 US disclosed
US-6482849-B1 Inhibitors of α4β1 mediated cell adhesion TANABE SEIYAKU CO., LTD. (JP) 2002-11-19 US disclosed