SCHEMBL7106083

SCHEMBL7106083

COc1cccc(-c2cccc3[nH]nc(C4CCNCC4)c23)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.44
JAK3 P52333 1/20 0.44
PTK2 Q05397 1/20 0.44
JUND P17535 1/20 0.43
FOSB P53539 1/20 0.43
HTR2C P28335 2/20 0.43
HTR2A P28223 1/20 0.42
FYN P06241 2/20 0.41
HTR1A P08908 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
CCNT1 O60563 5/20 0.38
CDK9 P50750 5/20 0.38
TGFBR1 P36897 1/20 0.36
ACVR1 Q04771 1/20 0.36
MGAM O43451 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967919 0.76 JUND (0.39) JUNDFOSBHTR2CHTR2AHTR1A
SCHEMBL26811323 0.73 HTR2A (0.50) JUNDFOSBHTR2CHTR2A
SCHEMBL24330092 0.72 HTR1A (0.41) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL24329831 0.71 JUND (0.52) JUNDFOSBHTR2CFYNHTR1A
Hydrochloric Acid SCHEMBL26911829 0.70 HTR2C (0.51) JUNDFOSBHTR2CFYNHTR1A
SCHEMBL5584542 0.70 HTR2C (0.73) HTR2CHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL26811325 0.69 HTR2A (0.45) HTR2CHTR2ACCNT1CDK9
Acetic Acid SCHEMBL7965027 0.68 HTR2C (0.41) HTR2CFYN
SCHEMBL17837929 0.68 FYN (0.45) HTR2CFYNHTR1ASLC6A2SLC6A4
SCHEMBL196440 0.67 MGAM (0.55) MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355904-A2 HETEROCYCLINDAZOLE AND AZAINDAZOLE COMPOUNDS AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-10-29 EP disclosed
WO-2002051837-A2 HETEROCYCLINDAZOLE AND AZAINDAZOLE COMPOUNDS AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-07-04 WO disclosed