SCHEMBL7112013

SCHEMBL7112013

FC(F)(F)c1cccc(/C=C/Nc2ccccn2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.46
FBP1 P09467 1/20 0.43
P4HB P07237 1/20 0.43
PHGDH O43175 1/20 0.42
CTSC P53634 1/20 0.42
MEN1 O00255 2/20 0.42
LMNA P02545 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 2/20 0.42
HSP90AA1 P07900 1/20 0.42
PKM P14618 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.41
TLR7 Q9NYK1 1/20 0.40
MAPK1 P28482 1/20 0.40
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7112014 1.00 NFE2L2 (0.46) NFE2L2FBP1P4HBPHGDHCTSC
SCHEMBL4085102 0.78 NPC1 (0.54) MEN1LMNAKMT2AMAPTPKM
SCHEMBL4085100 0.78 NPC1 (0.54) MEN1LMNAKMT2AMAPTPKM
SCHEMBL715978 0.75 NFE2L2 (0.49) NFE2L2FBP1P4HBMEN1LMNA
SCHEMBL715979 0.75 NFE2L2 (0.49) NFE2L2FBP1P4HBMEN1LMNA
SCHEMBL4656669 0.72 CTSC (0.65) CTSCMEN1LMNAKMT2AMAPT
SCHEMBL30128849 0.72 CTSC (0.65) CTSCMEN1LMNAKMT2AMAPT
SCHEMBL3904046 0.71 NFE2L2 (0.73) NFE2L2FBP1P4HBMEN1LMNA
SCHEMBL5496405 0.71 NFE2L2 (0.73) NFE2L2FBP1P4HBMEN1LMNA
SCHEMBL13763536 0.71 NPC1 (0.59) MEN1KMT2AMAPTPKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1443926-A1 PYRIDINE DERIVATIVES AS NMDA-RECEPTOR SUBTYPE BLOCKERS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-11 EP disclosed
WO-2003037333-A1 PYRIDINE DERIVATIVES AS NMDA-RECEPTOR SUBTYPE BLOCKERS F. HOFFMANN-LA ROCHE AG (CH) 2003-05-08 WO disclosed