SCHEMBL7112425

SCHEMBL7112425

O=C(Cl)N(c1ccccc1)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.47
PTGIR P43119 2/20 0.46
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
GAA P10253 2/20 0.44
TSHR P16473 1/20 0.44
ALDH1A1 P00352 3/20 0.44
APP P05067 1/20 0.44
HCAR3 P49019 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
PKM P14618 1/20 0.42
PLOD2 O00469 1/20 0.42
NAPRT Q6XQN6 1/20 0.41
KCNN4 O15554 1/20 0.40
NAMPT P43490 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL9479075 0.87 NPSR1 (0.50) HTTNPSR1GAATSHRALDH1A1
SCHEMBL310005 0.82 NPSR1 (0.64) HTTNPSR1GAATSHRALDH1A1
SCHEMBL1648430 0.82 KCNA5 (0.47) KCNA5PTGIRHTTNPSR1GAA
SCHEMBL7982484 0.82 HTT (0.49) KCNA5PTGIRHTTNPSR1GAA
SCHEMBL16398787 0.81 GAA (0.50) KCNA5PTGIRHTTNPSR1GAA
Hydrochloric Acid SCHEMBL27470915 0.81 KCNA5 (0.46) KCNA5PTGIRHTTNPSR1GAA
SCHEMBL16295458 0.80 NOTUM (0.50) KCNA5HTTNPSR1GAATSHR
SCHEMBL17591716 0.79 HTT (0.56) KCNA5HTTGAATSHRALDH1A1
SCHEMBL28060972 0.76 HTT (0.50) KCNA5PTGIRHTTNPSR1GAA
SCHEMBL5633185 0.76 F7 (0.52) KCNA5PTGIRHTTGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1013639-B1 Aryl carboxylic acid and tetrazole derivatives comprising a carbamoyloxy unit HOFFMANN LA ROCHE (CH) 2003-10-01 EP disclosed
US-6335459-B1 PROSTAGLANDIN I2 RECEPTOR MODULATORS; TREATING TISSUE NECROSIS, PREMATURE UTERINE CONTRACTION, GASTRIC ULCERATION, SEXUAL DYSFUNCTION, MENSTRUAL PAIN AND IMPROPER WOUND HEALING, IMMUNOREGULATION, PLATELET AGGREGATION OR NEUTROPHIL FUNCTION SYNTEX (U.S.A.) LLC 2002-01-01 US disclosed
EP-1013639-A1 Aryl carboxylic acid and tetrazole derivatives comprising a carbamoyloxy unit F. HOFFMANN-LA ROCHE AG (CH) 2000-06-28 EP disclosed