SCHEMBL28060972

SCHEMBL28060972

CCNC(=O)N(c1ccccc1)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.50
GAA P10253 2/20 0.45
KCNA5 P22460 2/20 0.45
KCNN4 O15554 1/20 0.45
PTGIR P43119 1/20 0.44
PLOD2 O00469 1/20 0.44
KDM4E B2RXH2 1/20 0.44
HDAC6 Q9UBN7 2/20 0.43
TSHR P16473 1/20 0.43
NOTUM Q6P988 1/20 0.41
MAPT P10636 1/20 0.41
GFER P55789 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NPC1 O15118 2/20 0.41
PKM P14618 2/20 0.41
RAB9A P51151 2/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1400657 0.87 NPSR1 (0.50) HTTPTGIRTSHRNPSR1NPC1
SCHEMBL7982484 0.79 HTT (0.49) HTTGAAKCNA5KCNN4PTGIR
SCHEMBL11613500 0.79 CYP1A2 (0.61) HTTTSHRMAPTKMT2ASMN1; SMN2
SCHEMBL10855623 0.77 RECQL (0.41) HTTGAAMAPTGFERNPSR1
SCHEMBL1648430 0.76 KCNA5 (0.47) HTTGAAKCNA5KCNN4PTGIR
SCHEMBL7112425 0.76 KCNA5 (0.47) HTTGAAKCNA5KCNN4PTGIR
SCHEMBL966680 0.75 OPRM1 (0.51) HTTKDM4ETSHRNPC1PKM
SCHEMBL13266974 0.75 RIPK1 (0.60) PKMKMT2ASMN1; SMN2
SCHEMBL16398787 0.75 GAA (0.50) HTTGAAKCNA5KCNN4PTGIR
Hydrochloric Acid SCHEMBL27470915 0.74 KCNA5 (0.46) HTTGAAKCNA5KCNN4PTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102725290-B As the condensed heterocyclic compouds of ion channel modulators GILEAD SCIENCES, INC. (US) 2016-03-09 CN claimed
CN-102725290-B As the condensed heterocyclic compouds of ion channel modulators GILEAD SCIENCES, INC. (US) 2016-03-09 CN disclosed