SCHEMBL7118804

SCHEMBL7118804

O=C(O)N1C(=O)OC(c2ccc(Cl)nc2)C1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.39
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 1/20 0.38
GRM4 Q14833 1/20 0.38
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
KCNE1 P15382 2/20 0.38
KCNQ1 P51787 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
CETP P11597 1/20 0.35
CCR9 P51686 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CES2 O00748 1/20 0.34
MAOA P21397 1/20 0.34
FFAR2 O15552 1/20 0.34
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749376 0.87 KDM4E (0.37) CYP3A4KDM4EHSD17B10GRM4KCNQ3
SCHEMBL5751613 0.83 KCNN4 (0.39) KDM4ESMN1; SMN2ALDH1A1CES2LPL
SCHEMBL5752174 0.83 CES2 (0.37) SMN1; SMN2CES2SIRT2SIRT1
SCHEMBL5750077 0.81 CETP (0.38) CYP3A4CETP
SCHEMBL7116914 0.81 CES2 (0.34) KDM4EHSD17B10SMN1; SMN2ALDH1A1CES2
SCHEMBL5749040 0.75 CYP3A4 (0.38) CYP3A4KDM4EHSD17B10GRM4KCNQ3
SCHEMBL5749379 0.71 KDM4E (0.38) CYP3A4KDM4EHSD17B10GRM4KCNQ3
SCHEMBL6579476 0.70 KCNN4 (0.40) KDM4EALDH1A1
SCHEMBL5749152 0.70 MDM2 (0.37)
SCHEMBL5751187 0.69 EGLN2 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed