SCHEMBL711952

SCHEMBL711952

O=C(O)c1cccc(NS(=O)(=O)c2cccs2)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.67
KMT2A Q03164 5/20 0.67
HPGD P15428 2/20 0.63
ALDH1A1 P00352 3/20 0.63
POLB P06746 1/20 0.59
PFKFB3 Q16875 3/20 0.56
HTT P42858 1/20 0.55
HSD17B1 P14061 1/20 0.55
HSD17B2 P37059 1/20 0.55
BCHE P06276 1/20 0.54
HSD11B1 P28845 1/20 0.54
GAA P10253 2/20 0.53
KDM4E B2RXH2 1/20 0.52
TSHR P16473 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3563401 0.89 ALDH1A1 (0.67) MEN1KMT2AHPGDALDH1A1POLB
SCHEMBL27179624 0.87 BCHE (0.59) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL711991 0.85 HPGD (0.63) MEN1KMT2AHPGDALDH1A1POLB
SCHEMBL8266867 0.84 MEN1 (0.66) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL3563409 0.82 ALDH1A1 (0.66) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL3559462 0.82 LMNA (0.58) MEN1KMT2AHPGDALDH1A1
SCHEMBL27181100 0.80 MAPT (0.64) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL30926784 0.80 MAPT (0.64) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL4709087 0.80 MEN1 (0.84) MEN1KMT2AHPGDALDH1A1HTT
SCHEMBL29106437 0.79 ALDH1A1 (0.61) MEN1KMT2AHPGDALDH1A1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124617-B2 Imidazopyridine compounds TAKEDA SAN DIEGO, INC. (US) 2012-02-28 US disclosed
US-8124617-B2 Imidazopyridine compounds TAKEDA SAN DIEGO, INC. (US) 2012-02-28 US disclosed
US-8124617-B2 Imidazopyridine compounds TAKEDA SAN DIEGO, INC. (US) 2012-02-28 US disclosed
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS TAKEDA SAN DIEGO, INC. 2010-03-18 US disclosed
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS TAKEDA SAN DIEGO, INC. 2010-03-18 US disclosed
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS TAKEDA SAN DIEGO, INC. 2010-03-18 US disclosed
EP-1940837-A2 IMIDAZOPYRIDINE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2008-07-09 EP disclosed
WO-2007028135-A2 IMIDAZOPYRIDINE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed
WO-2007028135-A2 IMIDAZOPYRIDINE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed
WO-2005030709-A1 NOVEL SULFONE AMIDE DERIVATIVES CAPABLE OF INHIBITING BACE LG LIFE SCIENCES LTD. (KR) 2005-04-07 WO disclosed
US-4439444-A HISTAMINE RECEPTOR ANTAGONISTS SANOFI (FR) 1984-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069431-A1 IMIDAZOPYRIDINE COMPOUNDS GCK, GCKR, KHK MEN1 2868/4885KMT2A 2502/4885HPGD 727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.