SCHEMBL7121992

SCHEMBL7121992

CCOC(=O)CCC(C#N)(c1ccccc1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EBP Q15125 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
POLB P06746 1/20 0.45
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
KCNA3 P22001 1/20 0.39
OPRM1 P35372 1/20 0.39
PTPN1 P18031 1/20 0.38
ABCB1 P08183 1/20 0.38
PPID Q08752 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TOP2A P11388 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7315065 0.91 EBP (0.51) EBPSIGMAR1SMN1; SMN2POLBCYP4F2
SCHEMBL7120092 0.86 EBP (0.47) EBPSIGMAR1KCNA3ABCB1L3MBTL1
SCHEMBL5751980 0.83 EBP (0.51) EBPSIGMAR1SMN1; SMN2OPRM1L3MBTL1
SCHEMBL5230297 0.83 ABCB1 (0.40) EBPSIGMAR1SMN1; SMN2POLBCYP4F2
SCHEMBL5753399 0.82 EBP (0.50) EBPSIGMAR1SMN1; SMN2OPRM1L3MBTL1
SCHEMBL5752605 0.81 SIGMAR1 (0.47) EBPSIGMAR1CYP4F2CYP4A11OPRM1
SCHEMBL7826967 0.81 KCNA3 (0.52) SMN1; SMN2POLBCYP4F2CYP4A11KCNA3
SCHEMBL11845684 0.81 SMN1; SMN2 (0.50) EBPSIGMAR1SMN1; SMN2POLBCYP4F2
SCHEMBL5751743 0.80 KDM4E (0.40) CYP4F2CYP4A11L3MBTL1ALDH1A1
SCHEMBL29983875 0.80 POLB (0.51) SMN1; SMN2POLBCYP4F2CYP4A11KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US claimed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP claimed
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US disclosed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP disclosed