SCHEMBL5753399

SCHEMBL5753399

CC(=O)CCC(C#N)(c1ccccc1)C(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EBP Q15125 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
CYP2D6 P10635 5/20 0.39
CYP1A2 P05177 1/20 0.39
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C19 P33261 2/20 0.38
HIF1A Q16665 1/20 0.38
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
OPRM1 P35372 1/20 0.36
DRD3 P35462 1/20 0.36
KIF11 P52732 4/20 0.35
CHRM2 P08172 2/20 0.35
CHRM1 P11229 2/20 0.35
CHRM3 P20309 2/20 0.35
LMNA P02545 2/20 0.35
KCNH2 Q12809 1/20 0.35
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5751980 0.89 EBP (0.51) EBPSIGMAR1CYP2D6CYP1A2ALDH1A1
SCHEMBL5752605 0.84 SIGMAR1 (0.47) EBPSIGMAR1CYP2D6CYP1A2ALDH1A1
SCHEMBL7120092 0.84 EBP (0.47) EBPSIGMAR1CYP2D6CYP1A2ALDH1A1
SCHEMBL7304642 0.82 EBP (0.54) EBPSIGMAR1CYP2D6CYP1A2L3MBTL1
SCHEMBL7306091 0.82 EBP (0.54) EBPSIGMAR1CYP2D6CYP1A2L3MBTL1
SCHEMBL7121992 0.82 EBP (0.48) EBPSIGMAR1CYP2D6ALDH1A1L3MBTL1
SCHEMBL7753625 0.79 EBP (0.56) EBPSIGMAR1CYP2D6L3MBTL1CYP3A4
SCHEMBL5226760 0.79 EBP (0.56) EBPSIGMAR1CYP2D6CYP1A2L3MBTL1
SCHEMBL5237762 0.78 EBP (0.59) EBPSIGMAR1CYP2D6CYP1A2L3MBTL1
SCHEMBL7310593 0.77 EBP (0.51) EBPSIGMAR1CYP2D6CYP1A2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
CN-1310709-A N, N-substituted cyclic amine derivatives EISAI CO LTD (JP) 2001-08-29 CN disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed