SCHEMBL712371

SCHEMBL712371

C=CC(=O)OCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)C(C)(F)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 4/20 0.42
TP53 P04637 3/20 0.42
HIF1A Q16665 3/20 0.42
CYP3A4 P08684 2/20 0.42
HSD17B10 Q99714 1/20 0.42
THRB P10828 2/20 0.40
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL713578 1.00 TSHR (0.42) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL1321544 1.00 TSHR (0.42) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL709254 0.95 TSHR (0.43) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL30360186 0.90 TSHR (0.50) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL25869997 0.89 TSHR (0.43) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL14369078 0.89 TSHR (0.43) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL18085851 0.89 TSHR (0.43) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL18084881 0.89 TSHR (0.43) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL2462848 0.89 TSHR (0.46) TSHRHPGDALDH1A1TP53HIF1A
SCHEMBL44451 0.89 TSHR (0.46) TSHRHPGDALDH1A1TP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030194378-A1 Novel aerosol formulation containing a polar fluorinated molecule ASTRAZENECA AB (SE) 2003-10-16 US claimed
EP-1303258-A1 NOVEL AEROSOL FORMULATION CONTAINING A POLAR FLUORINATED MOLECULE AstraZeneca AB (SE) 2003-04-23 EP claimed
WO-2002003958-A1 NOVEL AEROSOL FORMULATION CONTAINING A POLAR FLUORINATED MOLECULE ASTRAZENECA AB (SE) 2002-01-17 WO claimed
US-11992367-B2 Acoustic-wave-probe resin material, acoustic lens, acoustic wave probe, acoustic wave determination device, ultrasound diagnostic apparatus, photo-acoustic wave determination device, ultrasonic endoscope, and method for producing acoustic lens FUJIFILM CORPORATION (JP) 2024-05-28 US disclosed
EP-3777696-B1 ACOUSTIC WAVE PROBE RESIN MATERIAL, ACOUSTIC LENS, ACOUSTIC WAVE PROBE, ACOUSTIC WAVE MEASURING APPARATUS, ULTRASONIC DIAGNOSTIC APPARATUS, PHOTOACOUSTIC WAVE MEASURING APPARATUS, ULTRASONIC ENDOSCOPE, AND METHOD FOR MANUFACTURING ACOUSTIC LENS FUJIFILM CORP (JP) 2024-02-28 EP disclosed
WO-2024024501-A1 POSITIVE PHOTOSENSITIVE RESIN COMPOSITION 日産化学株式会社 2024-02-01 WO disclosed
WO-2024024502-A1 POSITIVE-TYPE PHOTOSENSITIVE RESIN COMPOSITION 日産化学株式会社 2024-02-01 WO disclosed
US-11156750-B2 Laminated diffractive optical element and method for manufacturing laminated diffractive optical element CANON KABUSHIKI KAISHA (JP) 2021-10-26 US disclosed
US-11072707-B2 Resin material for acoustic wave probe, acoustic lens, acoustic wave probe, acoustic wave measurement apparatus, ultrasonic diagnostic apparatus, photoacoustic wave measurement apparatus, and ultrasound endoscope FUJIFILM CORPORATION (JP) 2021-07-27 US disclosed
US-20210223437-A1 OPTICAL ELEMENT AND METHOD FOR MANUFACTURING THE SAME CANON KK (JP) 2021-07-22 US disclosed
US-10996375-B2 Optical element and method for manufacturing the same CANON KABUSHIKI KAISHA (JP) 2021-05-04 US disclosed
EP-0890601-B1 SURFACE MODIFIED FLUOROELASTOMER SEALING MATERIAL NIHON VALQUA KOGYO KK (JP) 2006-05-24 EP disclosed
WO-2005085297-A1 TELECHELIC POLYMERS CONTAINING REACTIVE FUNCTIONAL GROUPS PENN STATE RESEARCH FOUNDATION (US) 2005-09-15 WO disclosed
US-20050182208-A1 Telechelic polymers containing reactive functional groups THE PENN STATE RESEARCH FOUNDATION 2005-08-18 US disclosed
US-20030194378-A1 Novel aerosol formulation containing a polar fluorinated molecule ASTRAZENECA AB (SE) 2003-10-16 US disclosed
EP-1303258-A1 NOVEL AEROSOL FORMULATION CONTAINING A POLAR FLUORINATED MOLECULE AstraZeneca AB (SE) 2003-04-23 EP disclosed
WO-2002003958-A1 NOVEL AEROSOL FORMULATION CONTAINING A POLAR FLUORINATED MOLECULE ASTRAZENECA AB (SE) 2002-01-17 WO disclosed
US-6074698-A CONTACTING A TREATMENT LIQUID CONTAINING A MONOMER HAVING A DOUBLE BOND, A POLYMERIZATION INITIATOR AND A SOLVENT WITH A RUBBER BASE MATERIAL; AND HEATING SO THAT THE MONOMER IS POLYMERIZED NIPPON VALDUA INDUSTRIES, LTD. (JP) 2000-06-13 US disclosed
EP-0890601-A1 PROCESS FOR PRODUCING SURFACE-MODIFIED RUBBER, SURFACE-MODIFIED RUBBER, AND SEALING MATERIAL NIPPON VALQUA INDUSTRIES, LTD. (JP) 1999-01-13 EP disclosed
EP-0632059-A2 Interpenetrating networks from unsaturated monomers and thermosetting resins SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1995-01-04 EP disclosed