SCHEMBL7126294

SCHEMBL7126294

O=[C]NC(c1ccccn1)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 3/20 0.40
KCNA5 P22460 5/20 0.39
KCNE1 P15382 2/20 0.39
TSHR P16473 2/20 0.39
SCN8A Q9UQD0 1/20 0.39
S1PR2 O95136 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR3 Q99500 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3751751 0.89 SLC6A2 (0.52) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL3305482 0.81 SLC6A3 (0.41) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL6537851 0.81 CYP1A2 (0.42) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL7517110 0.76 SLC6A2 (0.52) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL4980374 0.72 SLC6A3 (0.48) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL8815913 0.72 SLC6A2 (0.48) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL7126297 0.72 SLC6A2 (0.44) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL9185638 0.71 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL2339352 0.71 S1PR2 (0.50) SLC6A3SLC6A2SLC6A4NPSR1KDM4E
SCHEMBL833118 0.69 CYP1A2 (0.46) SLC6A3SLC6A2SLC6A4NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed