SCHEMBL7126602

SCHEMBL7126602

O=C(Nc1ccc(Br)cc1)c1ccccc1NS(=O)(=O)c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.70
KMT2A Q03164 8/20 0.70
KDM4E B2RXH2 3/20 0.70
ALDH1A1 P00352 2/20 0.70
LMNA P02545 2/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
HPGD P15428 1/20 0.70
CRHBP P24387 1/20 0.70
CYP2C19 P33261 1/20 0.70
HTT P42858 1/20 0.70
CRHR2 Q13324 1/20 0.70
NOD2 Q9HC29 1/20 0.70
GPR27 Q9NS67 4/20 0.60
AVPR2 P30518 1/20 0.60
SLC10A2 Q12908 1/20 0.60
SLC10A1 Q14973 1/20 0.60
SLC10A6 Q3KNW5 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862888 0.91 MEN1 (0.66) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL6755857 0.90 KMT2A (0.74) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL23200293 0.90 KDM4E (0.67) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL7120319 0.90 SLC10A6 (0.76) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL6862988 0.86 MEN1 (0.77) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL7213183 0.85 SLC10A6 (0.73) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL16088703 0.83 HTT (0.70) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL17538582 0.83 MEN1 (0.65) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL7213023 0.83 SLC10A6 (0.73) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL7116008 0.82 SLC10A6 (0.85) MEN1KMT2AALDH1A1LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030216449-A1 Phosphate transport inhibitors SMITHKLINE BEECHAM CORPORATION 2003-11-20 US claimed
CN-1429108-A Phosphate transport inhibitors SMITHKLINE BEECHAM CORP (US) 2003-07-09 CN claimed
EP-1202729-A1 PHOSPHATE TRANSPORT INHIBITORS SmithKline Beecham Corporation (US) 2002-05-08 EP claimed
WO-2001087294-A1 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-11-22 WO claimed
WO-2001005398-A1 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-25 WO claimed
US-20030216449-A1 Phosphate transport inhibitors SMITHKLINE BEECHAM CORPORATION 2003-11-20 US disclosed
CN-1429108-A Phosphate transport inhibitors SMITHKLINE BEECHAM CORP (US) 2003-07-09 CN disclosed
EP-1202729-A1 PHOSPHATE TRANSPORT INHIBITORS SmithKline Beecham Corporation (US) 2002-05-08 EP disclosed
WO-2001087294-A1 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-11-22 WO disclosed
WO-2001005398-A1 PHOSPHATE TRANSPORT INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030216449-A1 Phosphate transport inhibitors SLC34A2, SLC34A1, SLC34A3 MEN1 3779/4885KMT2A 4033/4885KDM4E 2954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.