SCHEMBL7127093

SCHEMBL7127093

O=C(O)c1cn(CC2CCNCC2)c2cc(I)ccc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 3/20 0.42
BRD4 O60885 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
CYP2J2 P51589 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TOP1 P11387 3/20 0.40
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 1/20 0.38
APEX1 P27695 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CNR1 P21554 7/20 0.38
CNR2 P34972 6/20 0.38
TOP2A P11388 1/20 0.38
CYP2C9 P11712 1/20 0.38
TOP2B Q02880 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7127615 0.86 LMNA (0.44) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL2997864 0.85 TOP1 (0.43) KDM4ELMNAALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL1430267 0.84 TOP1 (0.43) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL4142276 0.82 KDM4E (0.47) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL3004410 0.79 FEN1 (0.41) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL28787968 0.79 FEN1 (0.41) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL4149301 0.77 KDM4E (0.57) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL7120330 0.77 LMNA (0.48) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL8913601 0.76 LMNA (0.46) KDM4ELMNAALDH1A1HPGDHSD17B10
SCHEMBL1993306 0.75 CNR1 (0.45) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed