SCHEMBL7127445

SCHEMBL7127445

C=Cc1c(F)cc2c(=O)c(C(=O)OCC)cn(C3CC3)c2c1F

nearest known ligand 0.80

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.62
KMT2A Q03164 1/20 0.51
TOP2A P11388 7/20 0.49
TOP2B Q02880 7/20 0.49
STAT3 P40763 1/20 0.47
KCNH2 Q12809 3/20 0.45
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115999 0.92 ADRB2 (0.60) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL10413931 0.90 ADRB2 (0.52) ADRB2TOP2ATOP2BKCNH2KDM4E
SCHEMBL2844967 0.89 ADRB2 (0.68) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL29492858 0.89 ADRB2 (0.68) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL10627001 0.87 ADRB2 (0.66) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL7599453 0.86 ADRB2 (0.65) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL9693055 0.86 ADRB2 (0.65) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL114733 0.86 ADRB2 (0.60) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL5704396 0.85 ADRB2 (0.64) ADRB2KMT2ATOP2ATOP2BSTAT3
SCHEMBL143605 0.85 ADRB2 (0.64) ADRB2KMT2ATOP2ATOP2BSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
US-4945160-A Preparation of certain 7-substituted quinolones WARNER-LAMBERT COMPANY (US) 1990-07-31 US disclosed