SCHEMBL7128002

SCHEMBL7128002

COc1ccc(C2(c3ccccc3F)C=Cc3c(ccc4ccccc34)O2)cc1OC

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 8/20 0.35
ABCG2 Q9UNQ0 4/20 0.35
ABCC1 P33527 3/20 0.35
ABCB1 P08183 2/20 0.35
BCHE P06276 2/20 0.33
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818669 0.92 MAPT (0.35) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL27501457 0.89 HIF1A (0.34) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL2400659 0.86 KDM4E (0.38) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL5097862 0.83 KDM4E (0.40) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL8782282 0.81 ALDH1A1 (0.34) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL7821439 0.81 NPC1 (0.37) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL1387752 0.81 NPC1 (0.35) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL3926851 0.80 DPP4 (0.36) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL2599683 0.80 ALDH1A1 (0.38) MAPTMEN1KMT2AKDM4ENPC1
SCHEMBL1387824 0.80 NPC1 (0.35) MAPTMEN1KMT2AKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613475-B1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES INC (US) 1998-01-07 EP claimed
EP-0613475-A4 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS. PPG INDUSTRIES INC (US) 1995-02-08 EP claimed
EP-0613475-A1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES, INC. (US) 1994-09-07 EP claimed
WO-1993010112-A1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES, INC. (US) 1993-05-27 WO claimed
US-5066818-A Lenses, plastic transparencies PPG INDUSTRIES, INC. (US) 1991-11-19 US claimed
EP-0628064-B2 PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL INC (US) 2003-12-10 EP disclosed
EP-0728315-B1 PHOTOCHROMIC COMPOSITIONS OF IMPROVED FATIGUE RESISTANCE PPG IND OHIO INC (US) 1999-12-22 EP disclosed
EP-0628064-B1 PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL INC (US) 1999-04-07 EP disclosed
EP-0613475-B1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES INC (US) 1998-01-07 EP disclosed
EP-0728315-A1 PHOTOCHROMIC COMPOSITIONS OF IMPROVED FATIGUE RESISTANCE PPG INDUSTRIES, INC. (US) 1996-08-28 EP disclosed
EP-0728315-A4 PHOTOCHROMIC COMPOSITIONS OF IMPROVED FATIGUE RESISTANCE PPG INDUSTRIES INC (US) 1995-11-23 EP disclosed
US-5391327-A Includes hindered amine ligth stabilizer and asymmetric diaryloxalamide light stabilizer TRANSITIONS OPTICAL, INC. (US) 1995-02-21 US disclosed
EP-0628064-A1 PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL, INC. (US) 1994-12-14 EP disclosed
US-5369158-A And polymer TRANSITIONS OPTICAL, INC. (US) 1994-11-29 US disclosed
EP-0613475-A1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES, INC. (US) 1994-09-07 EP disclosed
WO-1994008260-A1 PHOTOCHROMIC COMPOSITIONS OF IMPROVED FATIGUE RESISTANCE PPG INDUSTRIES, INC. (US) 1994-04-14 WO disclosed
WO-1993017071-A1 PHOTOCHROMIC NAPHTHOPYRANS PPG INDUSTRIES, INC. (US) 1993-09-02 WO disclosed
US-5238981-A PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL, INC. (US) 1993-08-24 US disclosed
WO-1993010112-A1 PHOTOCHROMIC NAPHTHOPYRAN COMPOUNDS PPG INDUSTRIES, INC. (US) 1993-05-27 WO disclosed
US-5066818-A Lenses, plastic transparencies PPG INDUSTRIES, INC. (US) 1991-11-19 US disclosed