SCHEMBL7129147

SCHEMBL7129147

O=C1c2cccc3cccc(c23)N1CCCC(F)(F)F

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.57
ALDH1A1 P00352 1/20 0.57
CASP1 P29466 1/20 0.57
MPI P34949 1/20 0.57
CACNA1B Q00975 1/20 0.57
APBA1 Q02410 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
HTR7 P34969 10/20 0.56
HTR1A P08908 9/20 0.56
DRD2 P14416 9/20 0.56
HTR2A P28223 9/20 0.56
HTR6 P50406 9/20 0.56
UBE2N P61088 2/20 0.53
LMNA P02545 1/20 0.53
ATM Q13315 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HEXA P06865 2/20 0.52
HEXB P07686 2/20 0.52
TDP1 Q9NUW8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7120133 0.91 HPGD (0.60) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL9720971 0.86 HPGD (0.70) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL9290276 0.82 ALDH1A1 (0.64) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL9290382 0.81 HEXA (0.64) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL7131251 0.81 ALDH1A1 (0.71) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL7127209 0.80 CYP1B1 (0.53) ALDH1A1LMNA
SCHEMBL24991893 0.79 HPGD (0.60) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL9720875 0.78 ALDH1A1 (0.68) HPGDALDH1A1CASP1MPICACNA1B
SCHEMBL5423024 0.78 CES1 (0.67) ALDH1A1
SCHEMBL7071975 0.77 ALDH1A1 (0.66) HPGDALDH1A1CASP1MPICACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667303-B1 Agonists for serotonin 5-hydroxytryptamine 2C(5HT2C) receptor; 6-(1,4-diazepan-1-yl)benzo(cd)indol-2(1H)-ones, 6-(1,4-diazepan-1-yl)acenaphthylen-1(2H)-ones, and 5-(1,4-diazepan-1-yl)- 2H-naphtho(1,8-cd)isothiazole-1,1-dioxides WYETH 2003-12-23 US disclosed