SCHEMBL7129158

SCHEMBL7129158

O=C1c2cccc3c(N4CCCN(CCCc5ccccc5)CC4)ccc(c23)N1CC1CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 5/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
RAB9A P51151 2/20 0.45
MAPK1 P28482 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
AVPR1A P37288 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
BRD1 O95696 1/20 0.44
TAF1 P21675 1/20 0.44
BRPF1 P55201 1/20 0.44
HTR7 P34969 3/20 0.43
HTR1A P08908 4/20 0.42
CHRNB2 P17787 2/20 0.42
CHRNB4 P30926 2/20 0.42
CHRNA3 P32297 2/20 0.42
CHRNA4 P43681 2/20 0.42
DRD2 P14416 2/20 0.42
HTR2A P28223 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7131242 0.95 CYP1B1 (0.47) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7128976 0.92 CYP1B1 (0.48) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7130468 0.89 BRD1 (0.49) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7124526 0.89 CYP1B1 (0.48) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7119987 0.89 HTR7 (0.50) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7123027 0.88 MEN1 (0.54) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7128510 0.87 MEN1 (0.53) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7131215 0.87 MEN1 (0.53) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7120096 0.87 CYP1B1 (0.54) CYP1B1MEN1KMT2ARAB9AMAPK1
SCHEMBL7130585 0.86 BRD1 (0.49) CYP1B1MEN1KMT2ARAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667303-B1 Agonists for serotonin 5-hydroxytryptamine 2C(5HT2C) receptor; 6-(1,4-diazepan-1-yl)benzo(cd)indol-2(1H)-ones, 6-(1,4-diazepan-1-yl)acenaphthylen-1(2H)-ones, and 5-(1,4-diazepan-1-yl)- 2H-naphtho(1,8-cd)isothiazole-1,1-dioxides WYETH 2003-12-23 US claimed