SCHEMBL7129305

SCHEMBL7129305

COc1cc(C#N)cc(I)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.50
ALB P02768 1/20 0.50
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
CACNA1G O43497 1/20 0.39
CACNA1B Q00975 1/20 0.39
AR P10275 3/20 0.39
GPR35 Q9HC97 1/20 0.39
ACHE P22303 1/20 0.39
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
CA9 Q16790 1/20 0.38
GAK O14976 2/20 0.36
RIPK2 O43353 2/20 0.36
COQ8A Q8NI60 2/20 0.36
NLK Q9UBE8 2/20 0.36
PTGS2 P35354 1/20 0.35
CYP1A1 P04798 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10762528 0.88 TTR (0.58) TTRALBPDE4APDE4BPDE4C
SCHEMBL509507 0.86 ACHE (0.52) PDE4APDE4BPDE4CPDE4DCACNA1G
SCHEMBL18574315 0.84 TTR (0.43) TTRALBPDE4APDE4BPDE4C
SCHEMBL523729 0.78 AR (0.46) PDE4APDE4BPDE4CPDE4DCACNA1G
SCHEMBL524326 0.77 HPGD (0.44) PDE4APDE4BPDE4CPDE4DCACNA1G
SCHEMBL523635 0.77 TSHR (0.46) TTRALBPDE4APDE4BPDE4C
SCHEMBL9627301 0.74 AR (0.51) TTRALBARKDM4EALDH1A1
SCHEMBL6072170 0.74 AR (0.51) TTRALBCACNA1GCACNA1BAR
SCHEMBL31574687 0.73 PTGS2 (0.44) PDE4APDE4BPDE4CPDE4DCACNA1G
SCHEMBL31574689 0.73 PTGS2 (0.44) PDE4APDE4BPDE4CPDE4DCACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1136198-C Novel benzyl pyrimidines ��������ҩ�ɷ����޹�˾ 2004-01-28 CN disclosed
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
CN-1166831-A Novel benzyl pyrimidines HOFFMANN LA ROCHE (CH) 1997-12-03 CN disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed