SCHEMBL7129510

SCHEMBL7129510

COc1cccc(F)c1-c1nc2c([N+](=O)[O-])cccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.53
PKN2 Q16513 1/20 0.53
ADORA3 P0DMS8 1/20 0.48
MGAM O43451 2/20 0.48
GAA P10253 2/20 0.48
SI P14410 2/20 0.48
MGAM2 Q2M2H8 2/20 0.48
ALDH1A1 P00352 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
PARP1 P09874 3/20 0.43
DHODH Q02127 4/20 0.43
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
CBFB Q13951 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204856 0.88 PKN1 (0.63) PKN1PKN2ADORA3MGAMGAA
SCHEMBL4564392 0.82 MGAM (0.64) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7129517 0.81 TDP1 (0.43) ALDH1A1TDP1CYP3A4HPGDCYP2C19
SCHEMBL5202010 0.80 CBFB (0.58) MGAMGAASIMGAM2ALDH1A1
SCHEMBL8521677 0.79 CARM1 (0.41) MGAMGAASIMGAM2ALDH1A1
SCHEMBL9044494 0.77 MGAM (0.71) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7886398 0.76 PKN1 (0.73) PKN1PKN2ADORA3MGAMGAA
SCHEMBL8599658 0.76 PKN1 (0.56) PKN1PKN2ADORA3MGAMGAA
SCHEMBL27961282 0.72 PKN1 (0.79) PKN1PKN2ADORA3MGAMGAA
SCHEMBL28425038 0.71 TNKS (0.72) PKN1PKN2GAAALDH1A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0963371-B1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE US GOV HEALTH & HUMAN SERV (US) 2003-05-02 EP disclosed
EP-0963371-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-12-15 EP disclosed
WO-1998037072-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-08-27 WO disclosed