SCHEMBL7129517

SCHEMBL7129517

COc1cccc(F)c1-c1nc2cccc([N+](=O)[O-])c2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.40
AMY1A P0DUB6 3/20 0.40
RPS6KA2 Q15349 2/20 0.40
TNKS O95271 2/20 0.39
TNKS2 Q9H2K2 2/20 0.39
PARP2 Q9UGN5 2/20 0.39
MAPT P10636 3/20 0.37
PIN1 Q13526 2/20 0.37
GUSB P08236 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
APEX1 P27695 1/20 0.36
NOS3 P29474 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204870 0.88 MEN1 (0.43) TDP1ALDH1A1L3MBTL1MAPTGUSB
SCHEMBL7129510 0.81 PKN1 (0.53) TDP1ALDH1A1L3MBTL1AMY1ATNKS
SCHEMBL5202015 0.80 RPS6KA2 (0.45) AMY1ARPS6KA2MAPTGUSBNPC1
SCHEMBL9044504 0.77 GUSB (0.56) TDP1ALDH1A1L3MBTL1AMY1AMAPT
SCHEMBL2361351 0.73 AMY1A (0.45) ALDH1A1AMY1AMAPT
SCHEMBL1895139 0.72 MEN1 (0.56) TDP1ALDH1A1L3MBTL1TNKSTNKS2
SCHEMBL5771322 0.71 PARP1 (0.48) TDP1ALDH1A1L3MBTL1TNKSTNKS2
SCHEMBL1013587 0.71 MAPT (0.53) TDP1ALDH1A1L3MBTL1MAPTKDM4E
SCHEMBL7159716 0.70 ALDH1A1 (0.71) TDP1ALDH1A1L3MBTL1MAPTKDM4E
SCHEMBL13405986 0.70 NQO2 (0.46) ALDH1A1AMY1AMAPTGUSBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0963371-B1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE US GOV HEALTH & HUMAN SERV (US) 2003-05-02 EP disclosed
EP-0963371-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-12-15 EP disclosed
WO-1998037072-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-08-27 WO disclosed