SCHEMBL7129699

SCHEMBL7129699

O=C(NC(c1ccccn1)c1ccccn1)c1cccc(I)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
S1PR3 Q99500 9/20 0.55
S1PR4 O95977 6/20 0.55
S1PR2 O95136 4/20 0.55
F2 P00734 1/20 0.45
MTOR P42345 1/20 0.43
GRM5 P41594 1/20 0.43
MYC P01106 1/20 0.41
MAX P61244 1/20 0.41
S1PR1 P21453 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
KAT6A Q92794 1/20 0.40
GAA P10253 1/20 0.39
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
TP53BP1 Q12888 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19195652 0.77 S1PR3 (0.71) ALDH1A1S1PR3S1PR4S1PR2S1PR1
SCHEMBL12614850 0.77 S1PR3 (0.71) ALDH1A1S1PR3S1PR4S1PR2S1PR1
SCHEMBL1357366 0.73 GAA (0.56) ALDH1A1F2MTORGRM5HDAC1
SCHEMBL4875309 0.73 S1PR3 (0.50) ALDH1A1S1PR3S1PR4S1PR2S1PR1
SCHEMBL17680606 0.72 NPSR1 (0.59) F2MTORGRM5MYCMAX
SCHEMBL17018686 0.72 GRM5 (0.51) ALDH1A1F2MTORGRM5MYC
SCHEMBL2339352 0.72 S1PR2 (0.50) ALDH1A1S1PR3S1PR4S1PR2GAA
SCHEMBL19195494 0.71 S1PR3 (1.00) ALDH1A1S1PR3S1PR4S1PR2S1PR1
SCHEMBL27959751 0.71 S1PR2 (0.46) ALDH1A1S1PR3S1PR4S1PR2GAA
SCHEMBL28443884 0.70 HDAC1 (0.46) F2MTORGRM5MYCMAX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-B1 NOVEL BENZYL PYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-03-26 EP disclosed
US-5763450-A BACTERICIDES; TREATMENT OF INFECTIOUS DISEASES HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed