SCHEMBL7129850

SCHEMBL7129850

C=CC(N)Nc1cccc2c1C(=O)c1ccccc1C2=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.54
MAPK1 P28482 5/20 0.54
L3MBTL1 Q9Y468 5/20 0.54
EGFR P00533 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TDP1 Q9NUW8 2/20 0.54
RAB9A P51151 2/20 0.54
PABPC1 P11940 1/20 0.54
MAOA P21397 2/20 0.49
ADORA2A P29274 1/20 0.46
CYP1A2 P05177 3/20 0.43
ALDH1A1 P00352 5/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
POLB P06746 2/20 0.41
RAD52 P43351 2/20 0.41
GAA P10253 1/20 0.41
DNMT1 P26358 1/20 0.41
SMARCA2 P51531 1/20 0.41
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6438245 0.89 MAOA (0.41) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL10767796 0.84 MAOA (0.41) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL7122669 0.81 MAPT (0.54) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL10622198 0.81 MEN1 (0.54) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL30102541 0.79 MAPT (0.64) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL30102545 0.79 MAPT (0.64) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL6664436 0.76 MAPT (0.64) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL11585770 0.76 ADORA2A (0.50) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL126130 0.75 MAPT (0.58) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2
SCHEMBL9445880 0.75 MAPT (0.68) MAPTMAPK1L3MBTL1EGFRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030130272-A1 Anthracene derivatives as anti-cancer agents BTG INTERNATIONAL LIMITED (GB) 2003-07-10 US disclosed
EP-1244624-A1 ANTHRACENE DERIVATIVES AS ANTI-CANCER AGENTS BTG INTERNATIONAL LIMITED (GB) 2002-10-02 EP disclosed
WO-2001044190-A1 ANTHRACENE DERIVATIVES AS ANTI-CANCER AGENTS BTG INTERNATIONAL LIMITED (GB) 2001-06-21 WO disclosed
US-5935969-A Pyrido-thiopyrandoinazoles with antitumor activity UNIVERSITY OF VERMONT (US) 1999-08-10 US disclosed
US-5736523-A ADMINISTERING TO THE MAMMAL SUFFERING FROM CANCER BIOCHEM PHARMA INC. (CA) 1998-04-07 US disclosed
EP-0450021-B1 ANTI-CANCER COMPOUNDS BRITISH TECH GROUP (GB) 1994-02-02 EP disclosed
US-5132327-A ANTI-CANCER COMPOUNDS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1992-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130272-A1 Anthracene derivatives as anti-cancer agents TOP2B, TOP1, TOP2A MAPT 4884/4885MAPK1 3848/4885L3MBTL1 2430/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.